Therapy Matrix
Rx Only
Rx OnlyForm
capsules
Strength
100 mg
Pack
30 capsules
Breast Cancer
Inluriyo
imlunestrant · 100 mg
Efficacy Gauge · Clinical Signal
Target Engagement92%
Progression-Free Survival78%
Tolerability Profile84%
Mechanism of Action
Imlunestrant is an oral selective estrogen receptor degrader that drives complete degradation of the estrogen receptor, shutting down the ER signaling axis that fuels ER-positive tumor growth, including in tumors with ESR1 mutations.
Manufacturer
OncoVantaHealth
Target Protein
ER
Delivery
Tablets
Quantity
30 capsules
Critical Safety Information
Inluriyo is a prescription therapy. It may interact with CYP3A4 inhibitors and hormonal treatments. Do not co-administer with grapefruit. Report pregnancy or nursing status immediately. Requires ongoing hepatic monitoring.
Pricing Tier · Select Quantity
Total
$2,650
All orders require a valid prescription and clinical review before fulfillment. Final pricing confirmed after verification.
